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    Efficacy of DA-7218, a new oxazolidinone prodrug, in the treatment of experimental actinomycetoma produced by nocardia brasiliensis by Espinoza González, Nelly Alejandra, Welsh Lozano, Oliverio, De Torres, Noemi Waksman, Cavazos Rocha, Norma Cecilia, Ocampo Candiani, Jorge, Said Fernández, Salvador, Lozano Garza, Gerardo, Choi, Sung Hak, Vera Cabrera, Lucio

    Published 2008
    “…Two recently synthesized oxazolidinones: (R)-3-(4-(2-(2-methyltetrazol-5-yl)- pyridin-5-yl)-3-fluorophenyl)-5-hydroxymethyloxazolidin-2-one (DA-7157) and its corresponding pro-drug (R)-3-(4-(2-(2-methyltetrazol-5-yl)-pyridin-5-yl)-3-fluorophenyl)- 2-oxo-5-oxazolidinyl) methyl disodium phosphate (DA-7218), have shown very good activity against several Gram positive bacteria, including Nocardia and Mycobacterium. …”
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